
{"id":8066,"date":"2014-02-27T16:50:07","date_gmt":"2014-02-27T16:50:07","guid":{"rendered":"http:\/\/ibecbarcelona.eu\/new\/nanoparticules-com-a-transportadors-de-farmacs-anti-malaria\/"},"modified":"2015-01-08T09:01:35","modified_gmt":"2015-01-08T09:01:35","slug":"nanoparticules-com-a-transportadors-de-farmacs-anti-malaria","status":"publish","type":"post","link":"https:\/\/ibecbarcelona.eu\/ca\/nanoparticules-com-a-transportadors-de-farmacs-anti-malaria\/","title":{"rendered":"Nanopart\u00edcules com a transportadors de f\u00e0rmacs antimal\u00e0ria"},"content":{"rendered":"<p>L\u2019estudi, publicat al<em> Journal of Controlled Release<\/em>, indica que les nanopart\u00edcules s\u00f3n capaces de recon\u00e8ixer diferents esp\u00e8cies de <em>Plasmodium<\/em>. Aquest \u00e9s el seu major potencial com a transportadors de f\u00e0rmacs antimal\u00e0rics. <\/p>\n<p>Les ter\u00e0pies antimal\u00e0ria actuals requereixen d\u2019estrat\u00e8gies capaces d\u2019alliberar f\u00e0rmacs de manera selectiva en les c\u00e8l\u2022lules infectades de Plasmodium. En aquest estudi, els investigadors han explorat la utilitat de dos nanosistemes polim\u00e8rics, AGMA1 i ISA23, com a transportadors de f\u00e0rmacs antimal\u00e0rics quea ataquen selectivament al patogen. El primer, AGMA1, t\u00e9 tamb\u00e9 activitat antimal\u00e0rica. Cosa que ha estat demostrada <em>in vitro<\/em> per la inhibici\u00f3 en el creixement de <em>Plasmodium falciparum<\/em>.<\/p>\n<p>L\u2019estudi mostra que els dos pol\u00edmers s\u2019uneixen preferentment a les c\u00e8l\u2022lules sangu\u00ednies infectades per <em>Plasmodium<\/em>. A m\u00e9s a m\u00e9s, s\u00f3n capaces de recon\u00e8ixer esp\u00e8cies molt divergents de par\u00e0sits de la mal\u00e0ria, com <em>P. falciparum<\/em> i <em>P. yoelii<\/em>, que infecten a humans i a ratolins respectivament. L\u2019administraci\u00f3 de 0,8 mg\/kg de sals de cloroquina, tant de AGMA1 com de ISA23, van curar als ratolins infectats per <em>P.yoelii<\/em> mentre que els animals tractats amb ambd\u00f3s f\u00e0rmacs de forma lliure no van sobreviure.<\/p>\n<p>\u201cAquests pol\u00edmers que poden encapsular f\u00e0rmacs antimal\u00e0rics tenen una baixa toxicitat, son biodegradables i ataquen de forma selectiva als gl\u00f2buls vermells infectats per diferents esp\u00e8cies de <em>Plasmodium<\/em>\u201d, explica en Xavier Fern\u00e0ndez-Busquets, investigador principal del grup de Nanomal\u00e0ria de la unitat mixta IBEC\/CRESIB que va liderar l\u2019estudi. \u201cAix\u00f2 significa que els pol\u00edmers son candidats extremadament prometedors per a desenvolupar ter\u00e0pies antimal\u00e0ria.\u201d<\/p>\n<p>Aquest potencial existent ha estat impulsat per al finan\u00e7ament rebut de Fondazione Cariplo per a desenvolupar aquest prototips polim\u00e8rics amb l\u2019objectiu de dissenyar un nanovector antimal\u00e0ric preparat per entrar en els assajos precl\u00ednics. Aquest nanovector, al tractar-se d\u2019una ter\u00e0pia dirigida, ha estat dissenyat per transportar una dosi menor de f\u00e0rmac. Per aquest motiu \u00e9s possible que sigui l\u2019opci\u00f3 m\u00e9s econ\u00f2mica i viable per a l\u2019\u00c0frica.<\/p>\n<p><strong>Article de referencia:<\/strong><br \/>Urb\u00e1n P, Valle-Delgado JJ, Mauro N, Marques J, Manfredi A, Rottmann M, Ranucci E, Ferruti P, Fern\u00e0ndez-Busquets X. <a href=\"http:\/\/www.sciencedirect.com\/science\/article\/pii\/S0168365913009747\" target=\"_blank\">Use of poly(amidoamine) drug conjugates for the delivery of antimalarials to Plasmodium<\/a>. J Control Release. 2014 Jan 7;177C:84-95.<\/p>\n","protected":false},"excerpt":{"rendered":"<h3><img decoding=\"async\" class=\"left size-full wp-image-8062 lazyload\" data-src=\"https:\/\/ibecbarcelona.eu\/wp-content\/uploads\/2014\/02\/nanocaps.jpg\" border=\"0\" width=\"340\" height=\"210\" data-srcset=\"https:\/\/ibecbarcelona.eu\/wp-content\/uploads\/2014\/02\/nanocaps.jpg 340w, https:\/\/ibecbarcelona.eu\/wp-content\/uploads\/2014\/02\/nanocaps-300x185.jpg 300w, https:\/\/ibecbarcelona.eu\/wp-content\/uploads\/2014\/02\/nanocaps-242x150.jpg 242w, https:\/\/ibecbarcelona.eu\/wp-content\/uploads\/2014\/02\/nanocaps-150x92.jpg 150w\" data-sizes=\"(max-width: 340px) 100vw, 340px\" src=\"data:image\/svg+xml;base64,PHN2ZyB3aWR0aD0iMSIgaGVpZ2h0PSIxIiB4bWxucz0iaHR0cDovL3d3dy53My5vcmcvMjAwMC9zdmciPjwvc3ZnPg==\" style=\"--smush-placeholder-width: 340px; --smush-placeholder-aspect-ratio: 340\/210;\" \/> Els f\u00e0rmacs dins de les nanoc\u00e0psules \u2018reconeixen\u2019 les c\u00e8l\u2022lules infectades pels diferents tipus de mal\u00e0ria i els permet frenar la resist\u00e8ncia<\/h3>\n<p>Un estudi dut a terme per investigadors del Institut de Bioenginyeria de Catalunya (IBEC) i el Centre de Recerca de Salut Internacional de Barcelona (CRESIB) demostra que el f\u00e0rmac encapsulat en nanopart\u00edcules \u2013 sals de cloroquina en pol\u00edmers de poliamidomina \u2013 \u00e9s significativament m\u00e9s efectiu quan \u00e9s alliberat <em>in vivo<\/em> que els f\u00e0rmacs lliures (no encapsulats) i pot ajudar a frenar la resist\u00e8ncia de f\u00e0rmacs.<\/p>\n","protected":false},"author":4,"featured_media":8062,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[96],"tags":[],"post_formats":[],"class_list":["post-8066","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-noticies-de-recerca"],"yoast_head":"<!-- This site is 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